The
Comparative
Reaction Solvent Research
at Gaylord
Chemical Company,
L.L.C.
systematically compares DMSO performance versus other common solvents
in commercially important reactions. Using established references from the
chemi-
cal literature, our scientists test reaction systems to ascertain the yield,
selectivity,
and reaction rates of DMSO versus other solvents.
Nucleophilic
Aromatic Substitution (S
N
Ar)
reactions
are essential tools for the
synthesis
of many pharmaceutical targets (quinolone antibiotics) and agricultural
products (dinitrophenyl ether herbicides). Addition-elimination reactions
of this type
benefit from the use of dipolar aprotic solvents, and DMSO has been shown
to excel
as a reaction solvent in these applications.
Gaylord
Chemical Company's
Comparative
Reaction Solvent Research
Examines
Nucleophilic Aromatic Substitution
Gaylord
Chemical Company,
L.L.C. (GCC) is the world's
leading provider of Dimethyl
Sulfoxide (DMSO) solutions.
Beginning in the early
1960's ,GCC has been dedi-
cated to the development of
new uses for DMSO. In or-
der to meet customer-specific
needs, GCC has pioneered
the development of multiple
grades of DMSO, including
DMSO USP.
Gaylord Chemical's solutions
-based approach has contrib-
uted to the development and
growth of industries including
pharmaceuticals, hydro-
carbons, electronics, poly-
mers, coatings, agricultural
chemicals, and industrial
cleaners.
Gaylord Chemical's head-
quarters are located in Slidell,
Louisiana with manufactur-
ing, research, and develop-
ment facilities in nearby
Bogalusa, Louisiana. GCC
remains the only producer of
DMSO in the Western Hemi-
sphere.
D M
S O
DMSO
PRODUCT INFORMATION BULLETIN
dimethyl
sulfoxide
and the S
N
Ar
reaction
NO
2
Cl
O
2
N
NH
2
O
NH
2
HO
solvent
0
10
20
30
40
50
60
70
80
90
100
0
50
100
150
200
time
(min)
y
i
e
l
d
(
%
)
DMSO
NMP
DMF
An unusual
degree of
selectivity
was
seen in the reaction shown.
Excellent
yield
of
the
diphenyl ether product was obtained, even when a bifunctional nucleophile
was
employed.
NMP
and DMF produced product mixtures containing the corresponding diphenyl-
amine as a significant impurity.
Bulletin
153B
Oct
2007
Gaylord
Chemical Company, L.L.C.
Your
Global Leader For DMSO Solutions!
P.O.
Box 1209
Slidell,
LA 70459-1209 USA
1.800.426.6620
Office
1.985.649.0068
Fax
info@gaylordchemical.com